Medicinal Chemistry
IUPAC Recommendations
and Technical Reports
Lectures presented at the Polish-Austrian-German-Hungarian-Italian
Joint Meeting on Medicinal Chemistry, Kraków, Poland, 15-18 October
2003
Preface, K. Kiec-Kononowicz and B. Malawska
Predicting drug metabolism: Concepts and challenges
B. Testa, A.-L. Balmat, and A. Long
p. 907 [Abstract] [full
text - pdf 203KB]
Prion protein as a target for therapeutic interventions
P. P. Liberski
p. 915 [Abstract] [full
text - pdf 176KB]
Structural basis for 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic
acid (AMPA) receptor activation
T. N. Johansen, J. R. Greenwood, S. B. Vogensen, and P. Krogsgaard-Larsen
p. 921 [Abstract] [full
text - pdf 456KB]
Search for noncompetitive 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic
acid receptor (AMPAR) antagonists: Synthesis, pharmacological properties,
and computational studies
A. Chimirri, G. De Sarro, S. Quartarone, M. L. Barreca, R. Caruso,
L. De Luca, and R. Gitto
p. 931 [Abstract] [full
text - pdf 382KB]
Neuropeptide mimetics for pain management
A. W. Lipkowski, A. Misicka, D. B. Carr, G. Ronsisvalle, D. Kosson,
and I. Maszczynska Bonney
p. 941 [Abstract] [full
text - pdf 281KB]
New endomorphin analogs with mu-agonist and delta-antagonist properties
G. T�th, A. Keresztes, Cs. T�mb�ly, A. P�ter, F. F�l�p, D. Tourw�,
E. Navratilova, �. Varga, W. R. Roeske, H. I. Yamamura, M. Szucs, and
A. Borsodi
p. 951 [Abstract] [full
text - pdf 209KB]
Spacer conformation in biologically active molecules
J. Karolak-Wojciechowska and A. Fruzinski
p. 959 [Abstract] [full
text - pdf 244KB]
Discovery of new anti-inflammatory agents
F. F�l�p, L. L�z�r, Z. Szakonyi, M. Pihlavisto, S. Alaranta, P.
J. Vainio, A. Juhakoski, A. Marjam�ki, and D. J. Smith
p. 965 [Abstract] [full
text - pdf 239KB]
NO donors: Focus on furoxan derivatives
A. Gasco, R. Fruttero, G. Sorba, A. Di Stilo, and R. Calvino
p. 973 [Abstract] [full
text - pdf 246KB]
Passive and catalytic antibodies and drug delivery
G. M. Blackburn, J. H. Rickard, S. Cesaro-Tadic, D. Lagos, A. Mekhalfia,
L. Partridge, and A. Pl�ckthun
p. 983 [Abstract] [full
text - pdf 255KB]
Virtual combinatorial chemistry and in silico screening: Efficient
tools for lead structure discovery?
T. Langer and G. Wolber
p. 991 [Abstract] [full
text - pdf 148KB]
Development of modulators of multidrug resistance: A pharmacoinformatic
approach
G. F. Ecker and P. Chiba
p. 997 [Abstract] [full
text - pdf 269KB]
Hindered nucleoside analogs as antiflaviviridae agents
S. Manfredini, A. Angusti, A. C. Veronese, E. Durini, S. Vertuani,
F. Nalin, N. Solaroli, S. Pricl, M. Ferrone, M. Mura, M. A. Piano, B.
Poddesu, A. Cadeddu, P. La Colla, and R. Loddo
p. 1007 [Abstract] [full
text - pdf 297KB]
Solid- and solution-phase synthesis of bioactive dihydropyrimidines
D. Dallinger, A. Stadler, and C. O. Kappe
p. 1017 [Abstract] [full
text - pdf 245KB]
Synthesis of naturally occurring o-heterocyclic compounds of biological
activity
S. Antus, K. Gul�csi, L. Juh�sz, L. Kiss, and T. Kurt�n
p. 1025 [Abstract] [full
text - pdf 299KB]
IUPAC Recommendations and Technical Reports
Glossary of terms used in toxciokinetics (IUPAC Recommendations 2003)
M. Nordberg, J. Duffus, and D. M. Templeton
p. 1033 [Abstract] [full
text - pdf 319KB]